SCHEMBL4693235

SCHEMBL4693235

CCC(CC(N)=O)C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
CCR5 P51681 9/20 0.37
CCL5 P13501 8/20 0.34
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695968 0.91 LMNA (0.44) LMNATSHRCCR5CCL5ALDH1A1
SCHEMBL4695866 0.87 CCR5 (0.36) CCR5CCL5ALDH1A1
SCHEMBL4696881 0.83 CCL5 (0.38) LMNATSHRCCR5CCL5ALDH1A1
SCHEMBL4692061 0.82 CCR5 (0.37) LMNACCR5CCL5ALDH1A1
SCHEMBL4695377 0.79 CCR5 (0.37) TSHRCCR5CCL5
SCHEMBL4695010 0.78 KMT2A (0.38) CCR5CCL5ALDH1A1
SCHEMBL4692781 0.78 PKM (0.36) LMNATSHRCCR5CCL5ALDH1A1
SCHEMBL4694111 0.78 KMT2A (0.34) CCR5ALDH1A1
SCHEMBL4694498 0.76 CCR5 (0.37) CCR5CCL5
SCHEMBL4691790 0.76 CCR5 (0.42) CCR5CCL5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed