SCHEMBL4695010

SCHEMBL4695010

CC(CC(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1)C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
CCR5 P51681 8/20 0.38
CCL5 P13501 5/20 0.38
MEN1 O00255 1/20 0.36
PIK3CD O00329 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695866 0.84 CCR5 (0.36) KMT2AALDH1A1GAACCR5CCL5
SCHEMBL4692061 0.84 CCR5 (0.37) ALDH1A1CCR5CCL5PIK3CDCYP2C19
SCHEMBL4695377 0.83 CCR5 (0.37) CCR5CCL5CYP2C9CYP2C19HDAC1
SCHEMBL4694111 0.81 KMT2A (0.34) KMT2AALDH1A1CCR5KDM4EHDAC1
SCHEMBL4696881 0.81 CCL5 (0.38) ALDH1A1CCR5CCL5
SCHEMBL4695087 0.80 CCR5 (0.34) CCR5CCL5
SCHEMBL4692781 0.80 PKM (0.36) KMT2AALDH1A1CCR5CCL5MEN1
SCHEMBL4690185 0.78 POLB (0.40) KMT2AALDH1A1CCR5CCL5POLB
SCHEMBL4693235 0.78 LMNA (0.40) ALDH1A1CCR5CCL5
SCHEMBL4694498 0.77 CCR5 (0.37) CCR5CCL5CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed