SCHEMBL4694262

SCHEMBL4694262

Cc1ccc(NC(=O)CCN2CC3CN(C(=O)c4c(C)nn(C)c4C)CC3C2)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
POLB P06746 1/20 0.47
TP53 P04637 2/20 0.44
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 2/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693150 0.89 TP53 (0.53) NPC1RAB9APOLBTP53ALDH1A1
SCHEMBL3283591 0.87 CCL5 (0.51)
SCHEMBL3281859 0.86 CCR5 (0.52) SMN1; SMN2TP53ALDH1A1KMT2ALMNA
SCHEMBL4694331 0.86 TP53 (0.47) SMN1; SMN2POLBTP53ALDH1A1KMT2A
SCHEMBL4690401 0.86 TP53 (0.47) SMN1; SMN2POLBTP53ALDH1A1KMT2A
SCHEMBL4694268 0.85 POLB (0.45) SMN1; SMN2NPC1RAB9APOLBALDH1A1
SCHEMBL3282221 0.85 CCR5 (0.51) SMN1; SMN2TP53ALDH1A1LMNATSHR
SCHEMBL4690123 0.85 MAPT (0.49) SMN1; SMN2TP53ALDH1A1KMT2ALMNA
SCHEMBL4691529 0.85 ALDH1A1 (0.51) SMN1; SMN2TP53ALDH1A1KMT2ALMNA
SCHEMBL4694302 0.84 MAPT (0.55) SMN1; SMN2NPC1RAB9APOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed