SCHEMBL4694629

SCHEMBL4694629

CCn1nc(C)cc1C(=O)N1CC2CN(CCCNc3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 3/20 0.40
HTT P42858 3/20 0.40
MAPT P10636 5/20 0.37
GAA P10253 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.35
GFER P55789 1/20 0.35
UBE2M P61081 1/20 0.35
DCUN1D1 Q96GG9 1/20 0.35
CCR2 P41597 1/20 0.35
KCNH2 Q12809 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694624 0.86 POLB (0.44) ALDH1A1KDM4EHTTMAPTSMN1; SMN2
SCHEMBL4690373 0.85 TSHR (0.41) ALDH1A1HTTMAPTGAASMN1; SMN2
SCHEMBL4692697 0.84 ALDH1A1 (0.41) ALDH1A1KDM4EHTTMAPTGAA
SCHEMBL4692813 0.83 MAPT (0.44) ALDH1A1HTTMAPTSMN1; SMN2LMNA
SCHEMBL4695974 0.82 ALDH1A1 (0.43) ALDH1A1KDM4EHTTMAPTGAA
SCHEMBL4695667 0.81 SMN1; SMN2 (0.43) ALDH1A1KDM4EHTTMAPTGAA
SCHEMBL14436612 0.81 ALDH1A1 (0.45) ALDH1A1KDM4EHTTMAPTGAA
SCHEMBL3281865 0.81 CCR5 (0.52) ALDH1A1HTTMAPTGAASMN1; SMN2
SCHEMBL4694337 0.81 CCR5 (0.43) ALDH1A1HTTMAPTGAASMN1; SMN2
SCHEMBL4691640 0.81 MAPT (0.54) ALDH1A1KDM4EHTTMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed