SCHEMBL4695904

SCHEMBL4695904

O=C(O)N1CC2CC1CN2C1CCc2cccc(Cl)c21

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.36
PARP1 P09874 7/20 0.35
OPRL1 P41146 2/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
NOTUM Q6P988 2/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
KCNH2 Q12809 1/20 0.32
P2RX7 Q99572 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3026821 0.80 NPY5R (0.42) PARP1LMNAHTT
SCHEMBL4696444 0.76 SRD5A1 (0.37) ALDH1A1HTT
SCHEMBL4751235 0.75 GRIN2B (0.43) OPRL1OPRM1OPRD1OPRK1NOTUM
SCHEMBL4695276 0.71 ALDH1A1 (0.38) ALDH1A1
SCHEMBL4126107 0.68 TSHR (0.47) NOTUMP2RX7
SCHEMBL2554310 0.66 HSD11B1 (0.31)
SCHEMBL4748618 0.64 DRD2 (0.36) KCNH2ALDH1A1HTT
SCHEMBL5036242 0.64 ATM (0.32)
SCHEMBL15129413 0.63 P2RX7 (0.42) PARP1NOTUMTAS1R3TAS1R1TAS1R2
SCHEMBL16395440 0.63 P2RX7 (0.42) PARP1NOTUMTAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910374-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-04-16 EP disclosed
WO-2007007069-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed