SCHEMBL4695963

SCHEMBL4695963

NC(=O)Oc1cc(F)c(C(=O)N2CC3CN(CC[CH]c4ccccc4)C[C@H]3C2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.39
HCRTR2 O43614 4/20 0.39
CCR5 P51681 14/20 0.38
CCL5 P13501 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694113 0.83 CHRNB2 (0.40) CCR5
SCHEMBL4690594 0.81 CCR5 (0.44) HCRTR1HCRTR2CCR5
SCHEMBL4693258 0.79 HCRTR1 (0.41) HCRTR1HCRTR2CCR5
SCHEMBL4691783 0.79 HCRTR1 (0.41) HCRTR1HCRTR2CCR5
SCHEMBL4693713 0.78 CCR5 (0.49) HCRTR1HCRTR2CCR5CCL5
SCHEMBL4696786 0.78 CCR5 (0.43) HCRTR1HCRTR2CCR5CCL5
SCHEMBL4691336 0.78 HRH4 (0.46)
SCHEMBL4694094 0.77 CHRNB2 (0.44) CCR5
SCHEMBL4691191 0.77 HCRTR1 (0.40) HCRTR1HCRTR2
SCHEMBL4695464 0.77 HCRTR1 (0.44) HCRTR1HCRTR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed