SCHEMBL4703330

SCHEMBL4703330

Cc1nsc(N(CC#N)[C@@H](CC(C)C)C(N)=O)c1-c1ccc(N2CCNCC2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.41
CTSS P25774 10/20 0.41
CTSB P07858 9/20 0.41
CTSK P43235 8/20 0.41
MAP2 P11137 2/20 0.38
ACVR1 Q04771 3/20 0.34
TGFBR1 P36897 2/20 0.34
BMPR1B O00238 1/20 0.34
BMPR1A P36894 1/20 0.34
ACVRL1 P37023 1/20 0.34
USP28 Q96RU2 1/20 0.33
USP25 Q9UHP3 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
CTSC P53634 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703250 0.89 CTSL (0.46) CTSLCTSSCTSBCTSKACVR1
SCHEMBL4703327 0.89 CTSL (0.46) CTSLCTSSCTSBCTSKACVR1
SCHEMBL4699905 0.80 CTSS (0.41) CTSLCTSSCTSBCTSKACVR1
SCHEMBL4701807 0.79 TGFBR1 (0.36) CTSLCTSSCTSBCTSKACVR1
SCHEMBL4703971 0.78 CTSS (0.37) CTSLCTSSCTSBCTSKACVR1
SCHEMBL4703631 0.78 CTSL (0.39) CTSLCTSSCTSBCTSK
SCHEMBL4702148 0.78 CTSS (0.40) CTSLCTSSCTSBCTSK
SCHEMBL4698971 0.78 CTSL (0.49) CTSLCTSSCTSBCTSKACVR1
SCHEMBL4701723 0.77 KDM4E (0.35) CTSLCTSSCTSBCTSK
SCHEMBL4703010 0.77 CTSS (0.37) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed