SCHEMBL4703631

SCHEMBL4703631

Cc1nsc(N(CC#N)[C@@H](CC(C)C)C(N)=O)c1-c1ccc(S(=O)(=O)N2CCNCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.39
CTSB P07858 5/20 0.39
CTSS P25774 5/20 0.39
ALDH1A1 P00352 2/20 0.36
IKBKB O14920 6/20 0.34
CHUK O15111 6/20 0.34
CTSK P43235 3/20 0.34
MAPT P10636 2/20 0.32
GAA P10253 2/20 0.32
CA12 O43570 1/20 0.32
ABL1 P00519 1/20 0.32
CA2 P00918 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MDM2 Q00987 1/20 0.32
SRC P12931 1/20 0.32
NAMPT P43490 1/20 0.32
F13A1 P00488 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703250 0.87 CTSL (0.46) CTSLCTSBCTSSCTSK
SCHEMBL4703327 0.87 CTSL (0.46) CTSLCTSBCTSSCTSK
SCHEMBL4701995 0.85 CTSK (0.37) CTSLCTSBCTSSCTSKCA2
SCHEMBL4702728 0.82 RORC (0.35) CTSLCTSBCTSSCTSKMAPT
SCHEMBL4701632 0.81 FNTA (0.34)
SCHEMBL4699525 0.80 CTSL (0.38) CTSLCTSBCTSSCTSK
SCHEMBL4703027 0.80 CTSK (0.31) CTSLCTSBCTSSCTSK
SCHEMBL4701807 0.79 TGFBR1 (0.36) CTSLCTSBCTSSALDH1A1CTSK
SCHEMBL4703330 0.78 CTSL (0.41) CTSLCTSBCTSSCTSK
SCHEMBL4701723 0.77 KDM4E (0.35) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed