SCHEMBL4704579

SCHEMBL4704579

CCC(=O)c1ccc2c(c1)CN(CCCSc1nnc(-c3ccccn3)n1C)CC2

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 14/20 0.59
KCNH2 Q12809 13/20 0.59
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
HTT P42858 2/20 0.51
PAX8 Q06710 1/20 0.51
TSHR P16473 1/20 0.51
ALDH1A1 P00352 2/20 0.49
MAPT P10636 1/20 0.49
DRD2 P14416 12/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701185 0.88 DRD3 (0.57) DRD3KCNH2ALDH1A1MAPTDRD2
SCHEMBL6191945 0.86 DRD3 (0.58) DRD3KCNH2DRD2
SCHEMBL4705988 0.83 DRD3 (0.44) DRD3KCNH2DRD2
SCHEMBL4705931 0.83 DRD3 (0.43) DRD3KCNH2ALDH1A1DRD2
SCHEMBL4702577 0.81 ALDH1A1 (0.57) DRD3KCNH2NPC1RAB9AHTT
SCHEMBL4705240 0.80 DRD3 (0.58) DRD3KCNH2ALDH1A1MAPTDRD2
Hydrochloric Acid SCHEMBL4861989 0.80 ALDH1A1 (0.56) DRD3KCNH2NPC1RAB9AHTT
SCHEMBL4387104 0.79 DRD3 (0.59) DRD3KCNH2ALDH1A1MAPTDRD2
SCHEMBL4701966 0.79 DRD3 (0.56) DRD3KCNH2TSHRALDH1A1MAPT
SCHEMBL4706365 0.79 DRD3 (0.57) DRD3KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7465744-B2 Triazole compounds and the therapeutic use thereof ABBOTT GMBH & CO. KG (DE) 2008-12-16 US disclosed
EP-1594861-B1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF ABBOTT GMBH & CO KG (DE) 2008-06-18 EP disclosed
US-20060241137-A1 Dopamine-D3-receptor antagonists/agonists; high selectivity, bioavailability and high cerebral availability; central nervous system diorders; 2-{3-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio]propyl}-7-propionyl-1,2,3,4-tetrahydroisoquinoline ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2006-10-26 US disclosed
EP-1594861-A1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF Abbott GmbH & Co. KG (DE) 2005-11-16 EP disclosed
WO-2004069830-A1 TRIAZOLE COMPOUNDS AND THE THERAPEUTIC USE THEREOF ABBOTT GMBH & CO. KG (DE) 2004-08-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060241137-A1 Dopamine-D3-receptor antagonists/agonists; high selectivity, bioavailability and high cerebral availability; central nervous system diorders; 2-{3-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio]propyl}-7-propionyl-1,2,3,4-tetrahydroisoquinoline DRD3, SLC6A3, ADORA3 DRD3 1/4885KCNH2 887/4885NPC1 1494/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.