SCHEMBL4705490

SCHEMBL4705490

Cc1nnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2N(C)C)n1Cc1ccc(F)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.36
GRM2 Q14416 1/20 0.35
CDC7 O00311 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 1/20 0.35
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
NR1I2 O75469 1/20 0.34
NR3C1 P04150 1/20 0.34
AR P10275 1/20 0.34
RXRA P19793 1/20 0.34
POLB P06746 1/20 0.34
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
KMT2A Q03164 2/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708287 0.89 ALDH1A1 (0.37) GRM2SMN1; SMN2MAPTCYP2C9CYP2C19
SCHEMBL14279261 0.88 P2RX7 (0.34) P2RX7GRM2CDC7LMNASMN1; SMN2
SCHEMBL4707108 0.84 P2RX7 (0.36) P2RX7SMN1; SMN2MAPTTP53
SCHEMBL4709715 0.84 CDC7 (0.43) P2RX7GRM2CDC7SMN1; SMN2NR1H2
SCHEMBL4707457 0.83 CDC7 (0.42) P2RX7GRM2CDC7LMNANR1H2
SCHEMBL4707397 0.83 P2RX7 (0.36) P2RX7GRM2LMNASMN1; SMN2MAPT
SCHEMBL4706503 0.81 P2RX7 (0.37) P2RX7SMN1; SMN2MAPTTSHRALDH1A1
SCHEMBL4707141 0.78 SMN1; SMN2 (0.34) GRM2SMN1; SMN2MAPTKMT2AHTT
SCHEMBL4705643 0.76 MAPT (0.45) P2RX7SMN1; SMN2MAPTPOLBTP53
SCHEMBL4706998 0.75 SLC16A3 (0.32) GRM2SMN1; SMN2MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed