SCHEMBL4707181

SCHEMBL4707181

Cc1cc(C(=O)c2ccccc2Cl)c(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2C)nn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 9/20 0.40
RORC P51449 5/20 0.40
TACR1 P25103 1/20 0.39
GAA P10253 2/20 0.37
KDM4E B2RXH2 2/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 1/20 0.35
PTGER4 P35408 1/20 0.34
P2RX1 P51575 1/20 0.34
P2RX4 Q99571 1/20 0.34
P2RX7 Q99572 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.34
CDC7 O00311 1/20 0.34
PLK4 O00444 1/20 0.34
MAPK13 O15264 1/20 0.34
PDPK1 O15530 1/20 0.34
DAPK3 O43293 1/20 0.34
DYRK3 O43781 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708690 0.89 RORB (0.40) RORBRORCTACR1GAAPTGER4
SCHEMBL4705944 0.89 TACR1 (0.39) RORBRORCTACR1GAAKDM4E
SCHEMBL4705502 0.88 RORB (0.39) RORBRORCTACR1GAAKDM4E
SCHEMBL4708285 0.88 CDC7 (0.38) RORBRORCTACR1GAACDC7
SCHEMBL4706783 0.87 RORB (0.38) RORBRORCTACR1GAAPTGER4
SCHEMBL4759328 0.87 RORB (0.43) RORBRORCTACR1GAAKDM4E
SCHEMBL4707207 0.86 RORB (0.40) RORBRORCTACR1GAAKDM4E
SCHEMBL4707706 0.85 IDH1 (0.42) RORBRORCTACR1PTGER4P2RX7
SCHEMBL4707926 0.84 P2RX7 (0.36) RORBRORCTACR1GAAP2RX7
SCHEMBL4705184 0.83 TACR1 (0.44) RORBRORCTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed