SCHEMBL4705529

SCHEMBL4705529

COC(=O)Oc1cc2ccc(OC)cc2n1CC#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.43
MTNR1B P49286 9/20 0.43
DYRK1A Q13627 2/20 0.41
MAOA P21397 1/20 0.41
CLK1 P49759 2/20 0.41
DYRK3 O43781 1/20 0.41
CLK2 P49760 1/20 0.41
CLK3 P49761 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK2 Q92630 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
DYRK4 Q9NR20 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
KDM2B Q8NHM5 1/20 0.40
CCR9 P51686 1/20 0.40
CCR2 P41597 1/20 0.40
MAPT P10636 5/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708326 0.81 MTNR1A (0.43) MTNR1AMTNR1BKDM4E
SCHEMBL5622754 0.80 MTNR1A (0.61) MTNR1AMTNR1BDYRK1AMAOACLK1
SCHEMBL14206927 0.76 DYRK1A (0.51) MTNR1AMTNR1BDYRK1AMAOACLK1
SCHEMBL4706772 0.76 MEN1 (0.39) CCR9MAPTSMN1; SMN2RXFP1KDM4E
SCHEMBL4705661 0.75 KDM4E (0.44) MTNR1AMTNR1BCCR2MAPTKDM4E
SCHEMBL2242465 0.75 MTNR1A (0.52) MTNR1AMTNR1BDYRK1AMAOACCR9
SCHEMBL4707304 0.69 CNR2 (0.42) CCR2MAPTSMN1; SMN2RXFP1KDM4E
SCHEMBL3817923 0.68 KDM4E (0.60) CCR9CCR2MAPTSMN1; SMN2KDM4E
SCHEMBL4705478 0.67 KDM4E (0.36) CCR9MAPTSMN1; SMN2KDM4ENPC1
SCHEMBL16246760 0.65 CA2 (0.51) MTNR1AMTNR1BCCR9CCR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1625129-B1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT BAYER HEALTHCARE AG (DE) 2008-03-05 EP disclosed