SCHEMBL4707304

SCHEMBL4707304

N#CCn1c(OC(=O)O)cc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.42
CCR2 P41597 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP1A2 P05177 3/20 0.40
ALDH1A1 P00352 7/20 0.40
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
KDM4E B2RXH2 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
POLB P06746 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
NPC1 O15118 2/20 0.36
HPGD P15428 1/20 0.36
DAO P14920 1/20 0.36
MAPK1 P28482 1/20 0.36
STAT3 P40763 1/20 0.36
HSP90AA1 P07900 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9666902 0.79 CCR2 (0.61) CNR2CCR2L3MBTL1ALDH1A1KMT2A
SCHEMBL2400013 0.78 CCR2 (0.63) CNR2CCR2L3MBTL1CYP1A2ALDH1A1
SCHEMBL9240559 0.75 ALDH1A1 (0.64) CCR2L3MBTL1CYP1A2ALDH1A1KMT2A
SCHEMBL24170706 0.74 CCR2 (0.47) CNR2CCR2L3MBTL1CYP1A2ALDH1A1
SCHEMBL7837255 0.73 MTNR1A (0.58) CNR2CCR2CYP1A2ALDH1A1KMT2A
SCHEMBL4198025 0.72 MCL1 (0.57) ALDH1A1KMT2AMEN1KDM4ENPC1
SCHEMBL9239991 0.72 CCR2 (0.67) CCR2MAPTSMN1; SMN2
SCHEMBL1392918 0.71 NOD2 (0.64) ALDH1A1KMT2AMEN1KDM4ERXFP1
SCHEMBL30585515 0.71 NOD2 (0.64) ALDH1A1KMT2AMEN1KDM4ERXFP1
SCHEMBL10289428 0.71 CYP1A2 (0.49) CNR2CCR2L3MBTL1CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1625129-B1 HETEROCYCLYL-SUBSTITUTED DIHYDROQUINAZOLINES AND USE THEREOF AS AN ANTIVIRAL AGENT BAYER HEALTHCARE AG (DE) 2008-03-05 EP disclosed