SCHEMBL4705879

SCHEMBL4705879

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2cccc(C(F)(F)F)c2)c1-c1cncnc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORB Q92753 8/20 0.42
RORC P51449 5/20 0.42
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.39
PTGER4 P35408 1/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
IDH1 O75874 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
GRM2 Q14416 1/20 0.36
NPBWR1 P48145 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27538912 0.94 RORB (0.44) RORBRORCHTTL3MBTL1POLB
SCHEMBL4705482 0.94 RORB (0.41) RORBRORCHTTL3MBTL1IDH1
SCHEMBL4707594 0.92 RORB (0.43) RORBRORCHTTL3MBTL1POLB
SCHEMBL4708122 0.91 RORB (0.39) RORBRORCIDH1GRM2
SCHEMBL4704941 0.88 RORB (0.40) RORBRORCTP53
SCHEMBL4708283 0.87 RORB (0.39) RORBRORCIDH1GRM2
SCHEMBL4707066 0.87 RORB (0.41) RORBRORCIDH1GRM2
SCHEMBL4708468 0.87 RORB (0.41) RORBRORCIDH1GRM2
SCHEMBL4706229 0.87 IDH1 (0.44) RORBRORCIDH1GRM2SMN1; SMN2
Tradipitant SCHEMBL29810017 0.85 RORB (0.42) RORBRORCIDH1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed