SCHEMBL4707066

SCHEMBL4707066

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2ccc(F)c(C(F)(F)F)c2)c1-c1cncnc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORB Q92753 5/20 0.41
GRM2 Q14416 1/20 0.35
RPS6KB1 P23443 1/20 0.34
IDH1 O75874 1/20 0.34
NTRK1 P04629 1/20 0.34
RORC P51449 3/20 0.34
VNN1 O95497 2/20 0.34
KCNN4 O15554 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN9A Q15858 1/20 0.33
P2RX7 Q99572 1/20 0.33
GRM4 Q14833 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705528 0.94 RORB (0.43) RORBGRM2RPS6KB1IDH1RORC
SCHEMBL4708480 0.92 RORB (0.42) RORBGRM2RPS6KB1IDH1RORC
SCHEMBL4705879 0.87 RORB (0.42) RORBGRM2IDH1RORC
SCHEMBL4705482 0.87 RORB (0.41) RORBGRM2IDH1RORCVNN1
SCHEMBL4708468 0.86 RORB (0.41) RORBGRM2IDH1NTRK1RORC
SCHEMBL4708122 0.86 RORB (0.39) RORBGRM2IDH1NTRK1RORC
SCHEMBL4705301 0.85 RORB (0.42) RORBGRM2RPS6KB1RORCKCNN4
SCHEMBL4708283 0.84 RORB (0.39) RORBGRM2IDH1RORCSCN5A
SCHEMBL4704941 0.84 RORB (0.40) RORBNTRK1RORCKCNN4P2RX7
SCHEMBL27538912 0.81 RORB (0.44) RORBIDH1RORCVNN1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed