SCHEMBL4704941

SCHEMBL4704941

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2cccc(OC(F)(F)F)c2)c1-c1cncnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 1/20 0.40
HSD17B13 Q7Z5P4 2/20 0.39
KCNN4 O15554 2/20 0.38
SLC16A3 O15427 1/20 0.37
SLC16A1 P53985 1/20 0.37
MCTS1 Q9ULC4 1/20 0.37
RORC P51449 1/20 0.36
DRD1 P21728 1/20 0.36
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
P2RX7 Q99572 1/20 0.36
CNR2 P34972 1/20 0.35
F2RL3 Q96RI0 1/20 0.35
CHRM5 P08912 1/20 0.35
SCD O00767 1/20 0.35
NTRK1 P04629 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707334 0.94 RORB (0.42) RORBHSD17B13KCNN4SLC16A3SLC16A1
SCHEMBL4706684 0.92 RORB (0.41) RORBHSD17B13KCNN4SLC16A3SLC16A1
SCHEMBL4705879 0.88 RORB (0.42) RORBRORCTP53
SCHEMBL4706958 0.86 RORB (0.42) RORBHSD17B13KCNN4SLC16A3SLC16A1
SCHEMBL4705482 0.85 RORB (0.41) RORBRORC
SCHEMBL4707066 0.84 RORB (0.41) RORBKCNN4RORCP2RX7NTRK1
SCHEMBL4708122 0.82 RORB (0.39) RORBRORCNTRK1
SCHEMBL27538912 0.82 RORB (0.44) RORBRORC
SCHEMBL4707594 0.80 RORB (0.43) RORBRORCTP53
SCHEMBL4708283 0.79 RORB (0.39) RORBRORCP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed