SCHEMBL470591

SCHEMBL470591

ON[C@H]1CN(Cc2ccccc2)C[C@@H]1c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
FUCA1 P04066 2/20 0.43
NPY5R Q15761 1/20 0.42
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
DRD4 P21917 1/20 0.40
S1PR1 P21453 3/20 0.40
CYP2D6 P10635 1/20 0.40
KDM1A O60341 1/20 0.40
EED O75530 1/20 0.39
S1PR5 Q9H228 1/20 0.39
NTRK1 P04629 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470753 0.80 KDM1A (0.55) FUCA1DRD2DRD3S1PR1KDM1A
SCHEMBL463076 0.79 KMT2A (0.47) SIGMAR1CYP3A4CYP2C9DRD2DRD3
SCHEMBL463075 0.79 KMT2A (0.47) SIGMAR1CYP3A4CYP2C9DRD2DRD3
SCHEMBL470646 0.75 DRD2 (0.45) SIGMAR1FUCA1DRD2DRD3S1PR1
SCHEMBL470519 0.73 DPP4 (0.48) SIGMAR1FUCA1DRD2DRD3KDM1A
SCHEMBL7216583 0.72 USP30 (0.53) SIGMAR1S1PR1S1PR5
SCHEMBL7216590 0.72 USP30 (0.53) SIGMAR1S1PR1S1PR5
SCHEMBL7216580 0.72 USP30 (0.53) SIGMAR1S1PR1S1PR5
SCHEMBL6422642 0.72 UBE2M (0.47) SIGMAR1CYP3A4CYP2C9FUCA1NPY5R
SCHEMBL13186825 0.71 DRD2 (0.53) SIGMAR1FUCA1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147951-A1 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS PROSIDION LIMITED (GB) 2011-12-01 WO disclosed