SCHEMBL470673

SCHEMBL470673

CCc1noc(N2CCC(C(C)Oc3cnc(Cl)nc3)[C@H](F)C2)n1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 0.31
GPR119 Q8TDV5 2/20 0.31
GPR183 P32249 1/20 0.31
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470787 0.77 GPR119 (0.32) GPR119GPR183KCNH2
SCHEMBL470537 0.77 GPR119 (0.39) OPRK1GPR119
SCHEMBL120997 0.77 GPR119 (0.34) OPRK1GPR119GPR183KCNH2
SCHEMBL146465 0.77 GPR119 (0.34) OPRK1GPR119GPR183KCNH2
SCHEMBL470585 0.75 GPR119 (0.35) GPR119GPR183KCNH2
SCHEMBL461635 0.74 GPR119 (0.44) OPRK1GPR119GPR183
SCHEMBL470686 0.72 GPR119 (0.40) GPR119GPR183KCNH2
SCHEMBL470680 0.71 ALOX5AP (0.39) GPR119GPR183KCNH2
SCHEMBL461248 0.71 GPR119 (0.45) GPR119GPR183KCNH2
SCHEMBL461247 0.71 GPR119 (0.45) GPR119GPR183KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147951-A1 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS PROSIDION LIMITED (GB) 2011-12-01 WO disclosed