SCHEMBL4706783

SCHEMBL4706783

Cc1cc(C(=O)c2ccccc2Cl)c(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2ccncc2)nn1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORB Q92753 9/20 0.38
RORC P51449 5/20 0.38
TACR1 P25103 1/20 0.35
MAPK1 P28482 1/20 0.35
GRM2 Q14416 1/20 0.35
CDC7 O00311 1/20 0.34
PTGER4 P35408 1/20 0.34
IDH1 O75874 1/20 0.34
GAA P10253 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708690 0.94 RORB (0.40) RORBRORCTACR1CDC7PTGER4
SCHEMBL4707706 0.91 IDH1 (0.42) RORBRORCTACR1PTGER4IDH1
SCHEMBL4707207 0.91 RORB (0.40) RORBRORCTACR1GRM2PTGER4
SCHEMBL4708209 0.88 RORB (0.39) RORBRORCTACR1MAPK1GRM2
Tradipitant SCHEMBL2898629 0.87 RORB (0.42) RORBRORCTACR1MAPK1GRM2
Tradipitant SCHEMBL29810017 0.87 RORB (0.42) RORBRORCTACR1MAPK1GRM2
SCHEMBL4707926 0.87 P2RX7 (0.36) RORBRORCTACR1IDH1GAA
SCHEMBL4708172 0.87 RORB (0.46) RORBRORCTACR1MAPK1GRM2
SCHEMBL4707181 0.87 RORB (0.40) RORBRORCTACR1MAPK1GRM2
SCHEMBL25479760 0.85 RORB (0.39) RORBRORCMAPK1GRM2CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed