SCHEMBL4707219

SCHEMBL4707219

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2cc(Cl)cc(Cl)c2)c1-c1ccncc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORB Q92753 1/20 0.48
MAPK1 P28482 1/20 0.39
TDO2 P48775 2/20 0.37
IDO1 P14902 2/20 0.37
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707264 0.91 RORB (0.49) RORBTDO2IDO1ALDH1A1
SCHEMBL4707224 0.91 RORB (0.44) RORBMAPK1TDO2IDO1CYP19A1
SCHEMBL28434941 0.91 RORB (0.44) RORBMAPK1IDO1ALDH1A1TSHR
Tradipitant SCHEMBL2898629 0.88 RORB (0.42) RORBMAPK1
Tradipitant SCHEMBL29810017 0.88 RORB (0.42) RORBMAPK1
SCHEMBL4708282 0.85 RORB (0.40) RORBMAPK1
SCHEMBL4708480 0.85 RORB (0.42) RORBMAPK1
SCHEMBL4707594 0.85 RORB (0.43) RORB
SCHEMBL25479760 0.85 RORB (0.39) RORBMAPK1
SCHEMBL4708736 0.84 RORB (0.49) RORBMAPK1TDO2IDO1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed