SCHEMBL4708480

SCHEMBL4708480

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2ccc(F)c(C(F)(F)F)c2)c1-c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORB Q92753 3/20 0.42
GRM4 Q14833 2/20 0.36
RPS6KB1 P23443 1/20 0.35
RORC P51449 2/20 0.35
KDR P35968 1/20 0.34
MAPK1 P28482 1/20 0.34
VNN1 O95497 1/20 0.34
KCNN4 O15554 1/20 0.34
GRM2 Q14416 1/20 0.34
CDC7 O00311 1/20 0.34
BLM P54132 1/20 0.34
WRN Q14191 1/20 0.34
IDH1 O75874 1/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705528 0.92 RORB (0.43) RORBRPS6KB1RORCVNN1GRM2
SCHEMBL4707066 0.92 RORB (0.41) RORBGRM4RPS6KB1RORCVNN1
SCHEMBL4707594 0.87 RORB (0.43) RORBRORCGRM2
SCHEMBL4705301 0.87 RORB (0.42) RORBGRM4RPS6KB1RORCKCNN4
Tradipitant SCHEMBL2898629 0.87 RORB (0.42) RORBRORCKDRMAPK1GRM2
Tradipitant SCHEMBL29810017 0.87 RORB (0.42) RORBRORCKDRMAPK1GRM2
SCHEMBL4706699 0.85 RORB (0.42) RORBRORCMAPK1GRM2CDC7
SCHEMBL4708282 0.85 RORB (0.40) RORBRORCKDRMAPK1GRM2
SCHEMBL4707219 0.85 RORB (0.48) RORBMAPK1
SCHEMBL28434941 0.84 RORB (0.44) RORBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1312136-C Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2007-04-25 CN disclosed