SCHEMBL4708736

SCHEMBL4708736

Cc1c(-c2ncccc2C(=O)c2ccccc2Cl)nnn1Cc1cc(Cl)cc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 2/20 0.49
JAK2 O60674 2/20 0.37
JAK1 P23458 1/20 0.37
TDO2 P48775 2/20 0.35
IDO1 P14902 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
MAPT P10636 2/20 0.35
RECQL P46063 1/20 0.35
CDC7 O00311 1/20 0.35
PLK4 O00444 1/20 0.35
MAPK13 O15264 1/20 0.35
PDPK1 O15530 1/20 0.35
DAPK3 O43293 1/20 0.35
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
RPS6KA5 O75582 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PRKCG P05129 1/20 0.35
CDK1 P06493 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705134 0.90 RORB (0.45) RORBJAK2JAK1TDO2IDO1
SCHEMBL4759328 0.88 RORB (0.43) RORBSMN1; SMN2P2RX7PTGDR2RORC
SCHEMBL4705301 0.84 RORB (0.42) RORBJAK2JAK1RPS6KB1P2RX7
SCHEMBL4708293 0.84 RORB (0.40) RORBP2RX7RORC
SCHEMBL4707219 0.84 RORB (0.48) RORBTDO2IDO1MAPK1CYP19A1
SCHEMBL4706973 0.84 RORB (0.44) RORBSMN1; SMN2MAPTP2RX7KMT2A
SCHEMBL4707264 0.83 RORB (0.49) RORBTDO2IDO1SMN1; SMN2VNN1
SCHEMBL4706958 0.82 RORB (0.42) RORBP2RX7RORCCYP2C9
SCHEMBL4709738 0.81 RORB (0.42) RORBRPS6KA3P2RX7PTGDR2RORC
SCHEMBL4707224 0.79 RORB (0.44) RORBTDO2IDO1SMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed