SCHEMBL4707264

SCHEMBL4707264

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2cc(Cl)cc(Cl)c2)c1-c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 1/20 0.49
VNN1 O95497 1/20 0.39
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
P2RX7 Q99572 6/20 0.38
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2B6 P20813 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
F2 P00734 1/20 0.37
IDH1 O75874 1/20 0.37
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4709776 0.91 RORB (0.45) RORBVNN1ALDH1A1L3MBTL1P2RX7
SCHEMBL4707219 0.91 RORB (0.48) RORBALDH1A1IDO1TDO2
SCHEMBL4706229 0.89 IDH1 (0.44) RORBVNN1SMN1; SMN2IDH1
SCHEMBL4705528 0.86 RORB (0.43) RORBVNN1ALDH1A1L3MBTL1P2RX7
SCHEMBL4706981 0.86 IDH1 (0.42) RORBVNN1CYP2D6CYP2C9CYP2C19
SCHEMBL27538912 0.86 RORB (0.44) RORBVNN1L3MBTL1POLBIDH1
SCHEMBL4707334 0.84 RORB (0.42) RORBVNN1IDH1
SCHEMBL4708736 0.83 RORB (0.49) RORBVNN1P2RX7CYP2C9CYP3A4
SCHEMBL4708752 0.83 RORB (0.43) RORBP2RX7SMN1; SMN2IDH1
SCHEMBL4707224 0.82 RORB (0.44) RORBP2RX7SMN1; SMN2IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed