SCHEMBL4707334

SCHEMBL4707334

O=C(c1ccccc1Cl)c1cccnc1-c1nnn(Cc2cccc(OC(F)(F)F)c2)c1-c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 1/20 0.42
HSD17B13 Q7Z5P4 1/20 0.39
KCNA5 P22460 1/20 0.39
KCNH2 Q12809 1/20 0.39
DYRK1A Q13627 1/20 0.39
CHRM5 P08912 2/20 0.39
SLC16A3 O15427 1/20 0.39
SLC16A1 P53985 1/20 0.39
MCTS1 Q9ULC4 1/20 0.39
CYP11B1 P15538 3/20 0.39
CYP11B2 P19099 3/20 0.39
KCNN4 O15554 1/20 0.38
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
IDH1 O75874 1/20 0.37
RORC P51449 1/20 0.36
NPY5R Q15761 1/20 0.36
ABL1 P00519 1/20 0.36
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4704941 0.94 RORB (0.40) RORBHSD17B13CHRM5SLC16A3SLC16A1
SCHEMBL4706684 0.92 RORB (0.41) RORBHSD17B13CHRM5SLC16A3SLC16A1
SCHEMBL27538912 0.88 RORB (0.44) RORBIDH1RORCVNN1
SCHEMBL4706958 0.86 RORB (0.42) RORBHSD17B13KCNH2SLC16A3SLC16A1
SCHEMBL4706229 0.85 IDH1 (0.44) RORBIDH1RORCVNN1
SCHEMBL4705528 0.84 RORB (0.43) RORBIDH1RORCVNN1
SCHEMBL4707264 0.84 RORB (0.49) RORBIDH1VNN1
SCHEMBL4706981 0.82 IDH1 (0.42) RORBIDH1RORCVNN1
SCHEMBL4709776 0.82 RORB (0.45) RORBIDH1VNN1
SCHEMBL4705879 0.82 RORB (0.42) RORBIDH1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1312136-C Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2007-04-25 CN disclosed