SCHEMBL4706958

SCHEMBL4706958

Cc1c(-c2ncccc2C(=O)c2ccccc2Cl)nnn1Cc1cccc(OC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORB Q92753 1/20 0.42
KCNN4 O15554 2/20 0.41
PPARG P37231 9/20 0.41
PPARA Q07869 6/20 0.41
DRD1 P21728 2/20 0.41
CYP2C9 P11712 1/20 0.41
EGFR P00533 1/20 0.41
CHRM4 P08173 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRA2A P08913 1/20 0.41
ALOX5 P09917 1/20 0.41
ADRB3 P13945 1/20 0.41
DRD2 P14416 1/20 0.41
ADRA2B P18089 1/20 0.41
CHRM3 P20309 1/20 0.41
TACR2 P21452 1/20 0.41
TBXA2R P21731 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
OPRM1 P35372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4706973 0.87 RORB (0.44) RORBPTGER4RORCP2RX7
SCHEMBL4706684 0.87 RORB (0.41) RORBKCNN4DRD1HSD17B13CNR2
SCHEMBL4704941 0.86 RORB (0.40) RORBKCNN4DRD1HSD17B13CNR2
SCHEMBL4707334 0.86 RORB (0.42) RORBKCNN4DRD1KCNH2HSD17B13
SCHEMBL4759328 0.83 RORB (0.43) RORBPTGER4RORCP2RX7
SCHEMBL4705301 0.82 RORB (0.42) RORBKCNN4CYP2C9RORCP2RX7
SCHEMBL4705134 0.82 RORB (0.45) RORBRORCP2RX7
SCHEMBL4708736 0.82 RORB (0.49) RORBCYP2C9RORCP2RX7
SCHEMBL4708293 0.80 RORB (0.40) RORBRORCP2RX7
SCHEMBL4709738 0.77 RORB (0.42) RORBSLC16A3SLC16A1MCTS1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed