SCHEMBL4710134

SCHEMBL4710134

CN(C)CCCC(=O)Nc1ccc(-c2nc(C(=O)Nc3ccc(-c4nc(C(=O)O)cs4)cc3)cs2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.54
MAPT P10636 5/20 0.53
ATM Q13315 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
NPY1R P25929 1/20 0.53
NPY2R P49146 1/20 0.53
LMNA P02545 3/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ROCK1 Q13464 1/20 0.48
ALDH1A1 P00352 2/20 0.48
HDAC3 O15379 4/20 0.48
HDAC1 Q13547 4/20 0.48
HDAC7 Q8WUI4 4/20 0.48
HDAC8 Q9BY41 4/20 0.48
HDAC6 Q9UBN7 4/20 0.48
MAPK1 P28482 1/20 0.47
LTA4H P09960 1/20 0.47
MAPKAPK2 P49137 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12582207 0.92 TDP1 (0.51) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL2030417 0.88 RAB9A (0.51) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL2026703 0.77 HDAC1 (0.45) MAPTHDAC3HDAC1HDAC7HDAC8
SCHEMBL3928031 0.73 ALDH1A1 (0.54) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL14499642 0.71 THRA (0.62) ALDH1A1LTA4H
SCHEMBL5786149 0.71 TDP1 (1.00) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL30807388 0.71 TDP1 (0.49) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL30620397 0.71 TDP1 (0.82) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL3931641 0.71 ALDH1A1 (0.61) TDP1MAPTATMNPSR1L3MBTL1
SCHEMBL12790096 0.71 TDP1 (0.82) TDP1MAPTATMNPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727808-B1 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS SPIROGEN LTD (GB) 2008-11-12 EP disclosed
EP-1727808-A2 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS Spirogen Limited (GB) 2006-12-06 EP disclosed
WO-2005085177-A2 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS SPIROGEN LIMITED (GB) 2005-09-15 WO disclosed