SCHEMBL4714410

SCHEMBL4714410

O=C1NCC(Cc2ccccc2)N1c1ccc(O)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.46
KDM4E B2RXH2 3/20 0.44
ATM Q13315 1/20 0.44
KMT2A Q03164 2/20 0.43
P4HB P07237 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
GAA P10253 1/20 0.41
MMP2 P08253 1/20 0.41
ESR1 P03372 3/20 0.40
ESR2 Q92731 3/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
NPC1L1 Q9UHC9 1/20 0.40
DRD4 P21917 1/20 0.39
PLCG1 P19174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16915091 0.87 MEN1 (0.44) KIF11KMT2AMAPTMMP2SLC6A2
SCHEMBL16915098 0.82 DAGLB (0.42) SLC6A2SLC6A4SLC6A3
SCHEMBL11092534 0.73 MAPT (0.46) KIF11KDM4ETDP1MAPTGAA
SCHEMBL8683030 0.72 ALOX5 (0.42) KMT2AGAA
SCHEMBL13986107 0.71 EHMT2 (0.46) KMT2AMAPTGAASLC6A2SLC6A4
SCHEMBL21010215 0.71 KDM4E (0.40) KDM4EATMMAPTSLC6A2SLC6A4
SCHEMBL15133223 0.70 HTR2C (0.52) KMT2ANPC1GAA
SCHEMBL3703267 0.69 HCRTR2 (0.42) ATMKMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL8415370 0.69 GAA (0.40) KDM4EKMT2ATDP1GAA
SCHEMBL4653392 0.67 CYP2D6 (0.36) KMT2ATDP1NPC1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957073-A2 MEDICINAL DRUG OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-08-20 EP disclosed
WO-2007066784-A2 DIARYLETHER DERIVATIVES AS ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-06-14 WO disclosed
EP-1773797-A2 AROMATIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-04-18 EP disclosed
WO-2006014012-A2 AROMATIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-02-09 WO disclosed