SCHEMBL3703267

SCHEMBL3703267

Cc1c(Br)cccc1N1C(=O)NCC1Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.42
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NR3C1 P04150 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15873785 0.84 JAK2 (0.34) HCRTR2
SCHEMBL16915091 0.76 MEN1 (0.44) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL4714410 0.69 KIF11 (0.46) SLC6A2SLC6A4SLC6A3KMT2AATM
SCHEMBL16915098 0.67 DAGLB (0.42) HCRTR2SLC6A2SLC6A4SLC6A3
SCHEMBL13986107 0.66 EHMT2 (0.46) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL6824233 0.65 MDM2 (0.42) KMT2AATM
SCHEMBL123282 0.64 P2RX7 (0.51) KMT2A
SCHEMBL21010215 0.63 KDM4E (0.40) SLC6A2SLC6A4SLC6A3ATM
SCHEMBL411437 0.63 MMP2 (0.49)
SCHEMBL15873874 0.62 P2RX7 (0.44) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391602-A1 CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS Bristol-Myers Squibb Company (US) 2011-12-07 EP disclosed
WO-2010080481-A1 CARBAZOLE CARBOXAMIDE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-07-15 WO disclosed