SCHEMBL4715224

SCHEMBL4715224

CCOC(=O)Oc1ccc(OCCCN(C)C)c(C#Cc2cc(C)cc(C)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
KDM4E B2RXH2 5/20 0.34
SYK P43405 1/20 0.34
LMNA P02545 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ATM Q13315 1/20 0.33
PTPN1 P18031 1/20 0.33
ESR1 P03372 3/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710572 0.90 THRA (0.37) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4717150 0.89 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2KDM4EESR1
SCHEMBL4714324 0.88 THRA (0.39) ALDH1A1CYP1A2CYP2D6CYP2C19THRA
SCHEMBL4714453 0.85 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL7349972 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4712830 0.75 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4715746 0.73 ALDH1A1 (0.44) ALDH1A1CYP1A2KDM4EESR1
SCHEMBL4712903 0.73 HPGD (0.41) ALDH1A1CYP1A2THRATHRBLMNA
SCHEMBL4710329 0.71 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19
SCHEMBL7348551 0.70 KDM4E (0.42) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998459-B1 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2008-04-23 EP claimed