SCHEMBL7349972

SCHEMBL7349972

Cc1cc(C)cc(C#Cc2nc(C(=O)O)ccc2OCCCN(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
SYK P43405 1/20 0.40
KDM4E B2RXH2 11/20 0.38
TDP1 Q9NUW8 3/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
FFAR1 O14842 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4714453 0.89 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL7348551 0.88 KDM4E (0.42) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4715224 0.81 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4715746 0.79 ALDH1A1 (0.44) ALDH1A1CYP1A2KDM4EHRH1
SCHEMBL4712830 0.79 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4712903 0.76 HPGD (0.41) ALDH1A1CYP1A2LMNAGAA
SCHEMBL4710329 0.74 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19FFAR1
SCHEMBL4711565 0.73 HTR1B (0.45) ALDH1A1SMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL4710338 0.73 CYP1A2 (0.41) ALDH1A1CYP1A2CYP2D6CYP2C19KDM4E
SCHEMBL4717150 0.72 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2KDM4EHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998459-A2 PYRIDINE DERIVATIVES Novartis AG (CH) 2000-05-10 EP claimed
WO-1999002497-A2 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 1999-01-21 WO claimed