SCHEMBL4716576

SCHEMBL4716576

CCN(c1ccc(OC)cc1)C1CN(C(=O)O)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
CHRM2 P08172 1/20 0.40
CHRM3 P20309 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
OPRM1 P35372 3/20 0.39
GAA P10253 3/20 0.38
KMT2A Q03164 3/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
KDM4E B2RXH2 1/20 0.38
OPRD1 P41143 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4714260 0.86 MEN1 (0.43) ALDH1A1SMN1; SMN2GAAKMT2ACHRNB2
SCHEMBL4716374 0.84 CCR5 (0.42) POLB
SCHEMBL4713689 0.84 SMN1; SMN2 (0.38) ALDH1A1HPGDCHRM2CHRM3SMN1; SMN2
SCHEMBL4713873 0.83 HRH3 (0.38) ALDH1A1SMN1; SMN2OPRM1KMT2AMEN1
SCHEMBL1574996 0.80 GRIN2B (0.57) ALDH1A1HPGDSMN1; SMN2KMT2ARAB9A
SCHEMBL4713356 0.80 ALDH1A1 (0.41) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL26131091 0.78 ALDH1A1 (0.44) ALDH1A1HPGDCHRM2CHRM3SMN1; SMN2
SCHEMBL4711851 0.77 HTT (0.43) ALDH1A1HPGDSMN1; SMN2GAAKMT2A
SCHEMBL27594337 0.77 CNR1 (0.41) ALDH1A1SMN1; SMN2GAAKDM4ERAB9A
SCHEMBL29027733 0.75 NR1I2 (0.37) ALDH1A1CHRM2CHRM3SMN1; SMN2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed