SCHEMBL4713356

SCHEMBL4713356

CCN(c1ccc(C#N)cc1)C1CN(C(=O)O)C1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
PGR P06401 2/20 0.40
CCR5 P51681 2/20 0.39
PDK2 Q15119 2/20 0.39
KDM1A O60341 5/20 0.38
SLC6A3 Q01959 1/20 0.38
USP30 Q70CQ3 3/20 0.37
MLYCD O95822 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
HCRTR2 O43614 1/20 0.36
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713689 0.83 SMN1; SMN2 (0.38) ALDH1A1CCR5
SCHEMBL21825043 0.82 AR (0.44) ALDH1A1PGRCCR5PDK2KDM1A
SCHEMBL4713873 0.82 HRH3 (0.38) ALDH1A1PGR
SCHEMBL4716576 0.80 ALDH1A1 (0.40) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL4714260 0.77 MEN1 (0.43) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL4711851 0.76 HTT (0.43) ALDH1A1
SCHEMBL4716374 0.75 CCR5 (0.42) CCR5HCRTR2
SCHEMBL21824810 0.75 JAK2 (0.47) ALDH1A1CCR5PDK2KDM1AAR
SCHEMBL154345 0.74 MAOA (0.42) ALDH1A1PGRSLC6A3
SCHEMBL4715539 0.73 ALDH1A1 (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed