SCHEMBL4713873

SCHEMBL4713873

CCN(c1ccc(F)cc1)C1CN(C(=O)O)C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
S1PR1 P21453 1/20 0.36
ALOX12 P18054 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
OPRM1 P35372 3/20 0.35
PGR P06401 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
AGTR2 P50052 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713689 0.87 SMN1; SMN2 (0.38) S1PR1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL4716576 0.83 ALDH1A1 (0.40) MEN1KMT2AOPRM1ALDH1A1SMN1; SMN2
SCHEMBL4714471 0.82 OXTR (0.38) PGRCYP2D6CYP2C9ALDH1A1
SCHEMBL4713356 0.82 ALDH1A1 (0.41) PGRALDH1A1
SCHEMBL4716374 0.81 CCR5 (0.42) HRH3TDP1
SCHEMBL4714260 0.81 MEN1 (0.43) MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4711851 0.80 HTT (0.43) HRH3MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL1575208 0.79 GRIN2B (0.54) KMT2AALDH1A1SMN1; SMN2
SCHEMBL4713625 0.79 CYP2D6 (0.38) MEN1KMT2APGRCYP2D6CYP2C9
SCHEMBL4710667 0.78 OPRM1 (0.38) OPRM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed