SCHEMBL4718481

SCHEMBL4718481

COC(=O)CC1CCN(C(=O)CBr)Cc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
NAMPT P43490 2/20 0.37
KDM4E B2RXH2 1/20 0.37
NOTUM Q6P988 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CACNA1G O43497 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790682 0.78 NPC1 (0.47) ALDH1A1MAPTNAMPTNPC1RAB9A
SCHEMBL4789373 0.78 DPP4 (0.48) ALDH1A1TAAR1KDM4E
SCHEMBL4790954 0.78 NAMPT (0.47) NAMPT
SCHEMBL1470470 0.76 MTNR1A (0.50) ALDH1A1
SCHEMBL4789524 0.75 RAB9A (0.59) ALDH1A1MAPTNAMPTNPC1RAB9A
SCHEMBL4791121 0.75 CACNA1G (0.47) TDP1NAMPTCACNA1G
SCHEMBL4714941 0.73 GRIN2B (0.39) NAMPT
SCHEMBL4760965 0.73 NAMPT (0.45) NAMPT
SCHEMBL15715850 0.72 MTNR1A (0.49)
SCHEMBL4715261 0.71 NAMPT (0.40) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216230-B1 FUSED CYCLOHEPTANE AND FUSED AZACYCLOHEPTANE COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR ANTAGONISTS AMGEN INC (US) 2008-04-23 EP disclosed
US-6514964-B1 Treating diseases, conditions or disorders mediated by integrin receptors, such as vitronectin and fibronectin receptors AMGEN INC. 2003-02-04 US disclosed