SCHEMBL4718971

SCHEMBL4718971

O=c1c(-c2cc(F)ccc2C(F)(F)F)ccc2n1CCC2

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.33
DPP4 P27487 1/20 0.33
TRPA1 O75762 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
KDM1A O60341 2/20 0.31
MAOA P21397 2/20 0.31
PER2 O15055 1/20 0.31
AR P10275 4/20 0.31
HSD11B1 P28845 1/20 0.31
TLR8 Q9NR97 1/20 0.31
PPARG P37231 1/20 0.31
RORC P51449 1/20 0.31
KMT2A Q03164 1/20 0.31
SRD5A1 P18405 1/20 0.31
LRRK2 Q5S007 1/20 0.30
SCN9A Q15858 1/20 0.30
EPHX2 P34913 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14102084 0.79 PDE3B (0.34) CHRM5TRPA1PDE3BPDE3AKDM1A
SCHEMBL4722184 0.79 PDE3B (0.33) CHRM5TRPA1PDE3BPDE3AKDM1A
Hydrochloric Acid SCHEMBL4765559 0.78 PDE3B (0.33) CHRM5DPP4TRPA1PDE3BPDE3A
SCHEMBL4723904 0.76 PDE3B (0.40) PDE3BPDE3APPARGRORCKMT2A
SCHEMBL4724319 0.73 PDE3B (0.36) PDE3BPDE3AKDM1AMAOAPPARG
SCHEMBL4721234 0.73 PDE3B (0.46) PDE3BPDE3APPARGRORCKMT2A
SCHEMBL4722680 0.72 WDR5 (0.35) PDE3BPDE3AHSD11B1TLR8PPARG
SCHEMBL21131387 0.71 TRPA1 (0.49) CHRM5TRPA1ARHSD11B1SCN9A
SCHEMBL30568360 0.71 TRPA1 (0.49) CHRM5TRPA1ARHSD11B1SCN9A
SCHEMBL22016195 0.67 SMN1; SMN2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed