SCHEMBL4721234

SCHEMBL4721234

COC(=O)c1cc(-c2cc(F)ccc2C(F)(F)F)c(=O)n2c1CCC2

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 8/20 0.46
PDE3A Q14432 8/20 0.46
PDK2 Q15119 1/20 0.37
ALDH1A1 P00352 3/20 0.36
PPARG P37231 1/20 0.36
RORC P51449 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
LMNA P02545 2/20 0.35
HTT P42858 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CFTR P13569 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723904 0.87 PDE3B (0.40) PDE3BPDE3APPARGRORCKMT2A
SCHEMBL4724319 0.80 PDE3B (0.36) PDE3BPDE3AALDH1A1PPARGRORC
SCHEMBL4722184 0.79 PDE3B (0.33) PDE3BPDE3APPARGRORCKMT2A
SCHEMBL14102084 0.79 PDE3B (0.34) PDE3BPDE3APPARGRORCKMT2A
SCHEMBL4722680 0.78 WDR5 (0.35) PDE3BPDE3APPARGRORCKMT2A
Hydrochloric Acid SCHEMBL4765559 0.78 PDE3B (0.33) PDE3BPDE3AALDH1A1PPARGRORC
SCHEMBL18796708 0.73 PDE3B (0.80) PDE3BPDE3AALDH1A1KMT2AMEN1
SCHEMBL29200214 0.73 ALDH1A1 (0.55) PDE3BPDE3APDK2ALDH1A1KMT2A
SCHEMBL4718971 0.73 CHRM5 (0.33) PDE3BPDE3APPARGRORCKMT2A
SCHEMBL18152850 0.72 MAPK1 (0.50) PDE3BPDE3AALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed