SCHEMBL4724319

SCHEMBL4724319

O=C(O)Nc1cc(-c2cc(F)ccc2C(F)(F)F)c(=O)n2c1CCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
KMT2A Q03164 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
APP P05067 3/20 0.35
PPARG P37231 3/20 0.34
RORC P51449 3/20 0.34
NTRK1 P04629 1/20 0.33
KDM1A O60341 2/20 0.33
MAOA P21397 2/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
WDR5 P61964 1/20 0.32
RBP4 P02753 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723904 0.84 PDE3B (0.40) PDE3BPDE3AKMT2APPARGRORC
SCHEMBL4721234 0.80 PDE3B (0.46) PDE3BPDE3AKMT2APPARGRORC
SCHEMBL14102084 0.80 PDE3B (0.34) PDE3BPDE3AKMT2APPARGRORC
SCHEMBL4722184 0.80 PDE3B (0.33) PDE3BPDE3AKMT2ANPC1RAB9A
Hydrochloric Acid SCHEMBL4765559 0.79 PDE3B (0.33) PDE3BPDE3AKMT2APPARGRORC
SCHEMBL4718971 0.73 CHRM5 (0.33) PDE3BPDE3AKMT2APPARGRORC
SCHEMBL4722680 0.73 WDR5 (0.35) PDE3BPDE3AKMT2APPARGRORC
SCHEMBL30568360 0.64 TRPA1 (0.49) POLBGAA
SCHEMBL21131387 0.64 TRPA1 (0.49) POLBGAA
SCHEMBL16438539 0.63 MAPT (0.41) KMT2APOLBALDH1A1MAPTRBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed