SCHEMBL4721770

SCHEMBL4721770

CCOC(=O)C(N)Cc1cc(C)c(Cl)c(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 5/20 0.38
THRA P10827 4/20 0.38
PPARG P37231 1/20 0.38
GPR35 Q9HC97 1/20 0.37
TPH1 P17752 2/20 0.36
SLC7A5 Q01650 1/20 0.35
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
MMP8 P22894 1/20 0.33
SLC15A1 P46059 1/20 0.33
SCN9A Q15858 1/20 0.33
CPB2 Q96IY4 1/20 0.33
LMNA P02545 1/20 0.33
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3311074 0.99 THRB (0.37) THRBTHRAPPARGGPR35TPH1
SCHEMBL10679766 0.82 THRB (0.46) THRBTHRAPPARGTPH1SLC7A5
SCHEMBL4717339 0.80 ALDH1A1 (0.42) THRBTHRATPH1SLC7A5MMP8
Hydrochloric Acid SCHEMBL3316938 0.79 TPH1 (0.42) THRBTHRATPH1SLC7A5MMP8
SCHEMBL5234664 0.79 CPB2 (0.40) THRBTHRATPH1SLC7A5CYP4F2
SCHEMBL4035263 0.78 TPH1 (0.42) THRBTHRAPPARGTPH1SLC7A5
SCHEMBL4035478 0.78 TPH1 (0.42) THRBTHRAPPARGTPH1SLC7A5
SCHEMBL3877275 0.78 TPH1 (0.42) THRBTHRAPPARGTPH1SLC7A5
SCHEMBL4717979 0.77 SMN1; SMN2 (0.43) TPH1SLC7A5CYP4F2CYP4A11
Hydrochloric Acid SCHEMBL3312834 0.76 SMN1; SMN2 (0.43) TPH1SLC7A5CYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP disclosed
EP-1558600-A1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-08-03 EP disclosed
WO-2004037810-A1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-05-06 WO disclosed