SCHEMBL4722181

SCHEMBL4722181

CCOC(=O)N1CCc2c(-c3cc(O)cc(O)c3)nn(-c3cc(N4CC[C@H](O)C4)ccc3C(F)(F)F)c(=O)c21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.36
RORC P51449 1/20 0.33
MYC P01106 2/20 0.32
WDR5 P61964 2/20 0.32
PDE3B Q13370 2/20 0.32
PDE3A Q14432 2/20 0.32
CXCR3 P49682 3/20 0.32
CACNA2D1 P54289 1/20 0.32
CACNA2D2 Q9NY47 1/20 0.32
NOTUM Q6P988 2/20 0.31
SOS1 Q07889 2/20 0.31
LGMN Q99538 1/20 0.31
HSD11B1 P28845 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722188 1.00 P2RX7 (0.36) P2RX7RORCMYCWDR5PDE3B
SCHEMBL4718551 0.92 P2RX7 (0.36) P2RX7CXCR3CACNA2D1CACNA2D2SOS1
SCHEMBL4718554 0.92 P2RX7 (0.36) P2RX7CXCR3CACNA2D1CACNA2D2SOS1
SCHEMBL14101734 0.90 ALDH1A1 (0.35) P2RX7CXCR3NOTUM
SCHEMBL4720220 0.88 F10 (0.35) P2RX7RORCCXCR3NOTUM
SCHEMBL4720216 0.88 F10 (0.35) P2RX7RORCCXCR3NOTUM
SCHEMBL4723006 0.85 P2RX7 (0.35) P2RX7PDE3BPDE3ASOS1HSD11B1
SCHEMBL4723010 0.85 P2RX7 (0.35) P2RX7PDE3BPDE3ASOS1HSD11B1
SCHEMBL4722245 0.84 P2RX7 (0.38) P2RX7RORCMYCWDR5PDE3B
SCHEMBL4722249 0.84 P2RX7 (0.38) P2RX7RORCMYCWDR5PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed