SCHEMBL4722667

SCHEMBL4722667

Cc1cc(C)cc(-c2nn(-c3cc(Br)ccc3C(F)(F)F)c(=O)c3c2CCN3CC(=O)O)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.34
CXCR3 P49682 1/20 0.32
AKR1B10 O60218 4/20 0.32
RET P07949 1/20 0.31
PRKX P51817 1/20 0.31
TAOK1 Q7L7X3 1/20 0.31
P2RX7 Q99572 1/20 0.31
NTRK1 P04629 1/20 0.31
AKR1B1 P15121 3/20 0.30
LMNA P02545 2/20 0.30
AKR1A1 P14550 1/20 0.30
XPO1 O14980 1/20 0.30
HPGD P15428 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TTR P02766 1/20 0.30
PTGER1 P34995 1/20 0.30
PMP22 Q01453 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
GFER P55789 1/20 0.30
GRIA1 P42261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14102047 0.91 AR (0.34) ARCXCR3RETPRKXTAOK1
SCHEMBL4720926 0.89 WDR5 (0.33) ARCXCR3AKR1B10RETPRKX
SCHEMBL4724885 0.81 SMPD3 (0.37)
SCHEMBL4724899 0.81 SMPD3 (0.37)
SCHEMBL4724015 0.81 MAPT (0.34) ARP2RX7NTRK1LMNANPSR1
SCHEMBL4722057 0.81 GRIN2B (0.35) AKR1B10P2RX7AKR1B1
SCHEMBL4723684 0.79 WDR5 (0.34) ARRETPRKXTAOK1
SCHEMBL14101709 0.78 F10 (0.39) CXCR3AKR1B10
SCHEMBL4720017 0.78 CXCR3 (0.31) CXCR3
SCHEMBL4721386 0.78 SMN1; SMN2 (0.33) RETPRKXTAOK1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed