SCHEMBL4725575

SCHEMBL4725575

C=CCN1C(=O)c2ccc(Cl)cc2C1=O

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.56
ALDH1A1 P00352 3/20 0.47
POLB P06746 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
S100A4 P26447 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
MEN1 O00255 1/20 0.42
CRHBP P24387 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
CRHR2 Q13324 1/20 0.42
ALDH2 P05091 1/20 0.40
GALR3 O60755 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26361645 0.82 CASP3 (0.59) CASP3ALDH1A1POLBRXFP1SMN1; SMN2
SCHEMBL31458661 0.82 CASP3 (0.53) CASP3ALDH1A1POLBRXFP1L3MBTL1
SCHEMBL7216276 0.80 S100A4 (0.47) ALDH1A1POLBS100A4MEN1KMT2A
SCHEMBL11045205 0.79 CASP3 (0.56) CASP3ALDH1A1POLBRXFP1SMN1; SMN2
SCHEMBL15046563 0.79 CASP3 (0.56) CASP3ALDH1A1POLBRXFP1SMN1; SMN2
SCHEMBL9778204 0.79 CASP3 (0.60) CASP3ALDH1A1POLBRXFP1SMN1; SMN2
SCHEMBL9244264 0.79 CASP3 (0.56) CASP3ALDH1A1POLBRXFP1L3MBTL1
SCHEMBL6827846 0.78 TDP1 (0.58) CASP3ALDH1A1POLBRXFP1SMN1; SMN2
SCHEMBL1547317 0.78 L3MBTL1 (0.53) CASP3ALDH1A1POLBRXFP1L3MBTL1
SCHEMBL170913 0.77 CASP3 (0.85) CASP3ALDH1A1POLBRXFP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108117645-B Method for preparing polyaryl imide and production device thereof 北京鼎益新材科技有限公司 2020-08-14 CN claimed
EP-1599438-B1 PREPARATION OF SUBSTITUTED PHTHALIC ANHYDRIDE, ESPECIALLY 4-CHLOROPHTALIC ANHYDRIDE GEN ELECTRIC (US) 2008-01-09 EP claimed
CN-1329360-C Preparation of substituted phthalic anhydride GEN ELECTRIC (US) 2007-08-01 CN claimed
CN-1751017-A Preparation of substituted phthalic anhydrides, especially 4-chlorophthalic anhydride GEN ELECTRIC (US) 2006-03-22 CN claimed
EP-1599438-A1 PREPARATION OF SUBSTITUTED PHTHALIC ANHYDRIDE, ESPECIALLY 4-CHLOROPHTALIC ANHYDRIDE GENERAL ELECTRIC COMPANY (US) 2005-11-30 EP claimed
EP-1458791-A1 METHODS FOR THE PREPARATION OF POLY(ETHERIMIDES)S GENERAL ELECTRIC COMPANY (US) 2004-09-22 EP claimed
WO-2004072012-A1 PREPARATION OF SUBSTITUTED PHTHALIC ANHYDRIDE, ESPECIALLY 4-CHLOROPHTALIC ANHYDRIDE GENERAL ELECTRIC COMPANY (A NEW YORK CORPORATION) (US) 2004-08-26 WO claimed
US-6590108-B1 Transimidation of bis(imide) in presence of phthalic anhydride having substituent selected from group consisting of nitro, bromo, fluoro and chloro, to yield dianhydride GENERAL ELECTRIC COMPANY 2003-07-08 US claimed
WO-2003050165-A1 METHODS FOR THE PREPARATION OF POLY(ETHERIMIDES)S GENERAL ELECTRIC COMPANY (US) 2003-06-19 WO claimed
US-6528663-B1 Transimidation between a substituted n-alkyl phthalimide and a substituted tetrahydrophthalic anhydride GENERAL ELECTRIC COMPANY 2003-03-04 US claimed
US-6498224-B1 SOLUTION POLYMERIZATION OF A DIANHYDRIDE AND A DIAMINE WHICH ELIMINATES THE NITRATION STEP; HIGH HEAT ENGINEERING PLASTICS GENERAL ELECTRIC COMPANY 2002-12-24 US claimed
CN-108117645-B Method for preparing polyaryl imide and production device thereof 北京鼎益新材科技有限公司 2020-08-14 CN disclosed