SCHEMBL7216276

SCHEMBL7216276

[CH2]CN1C(=O)c2ccc(Cl)cc2C1=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 2/20 0.47
PPOX P50336 1/20 0.42
ALDH1A1 P00352 3/20 0.41
ALDH2 P05091 2/20 0.41
ALDH3A1 P30838 2/20 0.41
KDM4E B2RXH2 4/20 0.41
NPC1 O15118 1/20 0.40
APAF1 O14727 1/20 0.39
CA9 Q16790 1/20 0.39
MEN1 O00255 2/20 0.38
HPGD P15428 2/20 0.38
KMT2A Q03164 2/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10451194 0.81 POLB (0.57) S100A4PPOXALDH1A1ALDH2ALDH3A1
SCHEMBL4725575 0.80 CASP3 (0.56) S100A4ALDH1A1ALDH2MEN1KMT2A
SCHEMBL6957475 0.79 CA9 (0.46) ALDH1A1KDM4EAPAF1CA9MEN1
SCHEMBL5878681 0.78 KDM4E (0.69) S100A4ALDH1A1KDM4ENPC1CA9
SCHEMBL10779928 0.78 KDM4E (0.46) S100A4ALDH1A1KDM4ENPC1MEN1
SCHEMBL1704408 0.78 S100A4 (0.52) S100A4PPOXALDH1A1ALDH2ALDH3A1
SCHEMBL6955085 0.77 CASP1 (0.55) S100A4ALDH1A1KDM4ENPC1APAF1
SCHEMBL6957181 0.77 PARK7 (0.45) KDM4ENPC1CA9
SCHEMBL522502 0.77 TDP1 (0.64) ALDH1A1KDM4ECA9MEN1HPGD
SCHEMBL4473721 0.77 ALDH1A1 (0.51) S100A4ALDH1A1KDM4ENPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095043-A1 TRIOXANE DERIVATIVES The Hong Kong University of Science & Technology (HK) 2001-05-02 EP claimed
WO-2000004026-A1 TRIOXANE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE & TECHNOLOGY (CN) 2000-01-27 WO claimed
EP-0974354-A1 Artemisinin derivatives The Hong Kong University of Science & Technology (HK) 2000-01-26 EP claimed
US-6649647-B1 Trioxane derivatives HAYNES RICHARD (CN) 2003-11-18 US disclosed
EP-1095043-A1 TRIOXANE DERIVATIVES The Hong Kong University of Science & Technology (HK) 2001-05-02 EP disclosed
WO-2000004026-A1 TRIOXANE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE & TECHNOLOGY (CN) 2000-01-27 WO disclosed
EP-0974354-A1 Artemisinin derivatives The Hong Kong University of Science & Technology (HK) 2000-01-26 EP disclosed