SCHEMBL4727326

SCHEMBL4727326

COc1ccnc(C2CC2C(=O)C23CC4CC(CC(C4)C2)C3)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
GRM1 Q13255 1/20 0.41
P2RX7 Q99572 1/20 0.41
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
P2RX2 Q9UBL9 1/20 0.40
LMNA P02545 1/20 0.40
ITK Q08881 1/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
FAAH O00519 1/20 0.39
CNR2 P34972 1/20 0.39
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8215134 0.86 ITK (0.35) KMT2AMEN1GRM1ALDH1A1KDM4E
SCHEMBL24737398 0.80 CCR1 (0.46) KMT2AMEN1KDM4ELMNAITK
SCHEMBL29302315 0.79 PLAU (0.47) KDM4ELMNAITKMAPTCCR1
SCHEMBL29302314 0.79 ITK (0.46) LMNAITKMAPTCCR1CCR5
SCHEMBL29879145 0.79 ITK (0.46) LMNAITKMAPTCCR1CCR5
SCHEMBL4731345 0.77 P2RX7 (0.49) KMT2AMEN1GRM1P2RX7ALDH1A1
Hydrochloric Acid SCHEMBL4728933 0.76 P2RX7 (0.48) KMT2AMEN1GRM1P2RX7ALDH1A1
SCHEMBL4729426 0.75 ALDH1A1 (0.49) KMT2AMEN1GRM1P2RX7ALDH1A1
SCHEMBL4728861 0.75 HPGDS (0.46) GRM1ITK
SCHEMBL24737400 0.75 NOS3 (0.46) KMT2AMEN1ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed