SCHEMBL4731345

SCHEMBL4731345

O=C(C1CC1c1ccccn1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.49
RAB9A P51151 3/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
AGTR1 P30556 1/20 0.48
OPRK1 P41145 1/20 0.48
RECQL P46063 1/20 0.48
GRM5 P41594 2/20 0.47
GRM1 Q13255 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
HSD11B1 P28845 2/20 0.46
ALDH1A1 P00352 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPK1 P28482 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4728933 0.99 P2RX7 (0.48) P2RX7RAB9AKDM4EMAPTAGTR1
SCHEMBL8215561 0.83 HSD11B1 (0.45) P2RX7RAB9AKDM4EMAPTAGTR1
SCHEMBL4731571 0.77 CNR1 (0.43) RAB9AKDM4EMAPTGRM1CYP3A4
SCHEMBL2518996 0.77 RIPK1 (0.48) RAB9AMAPTALDH1A1LMNAKMT2A
SCHEMBL13167851 0.77 RIPK1 (0.48) RAB9AMAPTALDH1A1LMNAKMT2A
SCHEMBL1207556 0.77 RIPK1 (0.48) RAB9AMAPTALDH1A1LMNAKMT2A
SCHEMBL29730159 0.77 RIPK1 (0.48) RAB9AMAPTALDH1A1LMNAKMT2A
SCHEMBL3596616 0.77 RIPK1 (0.48) RAB9AMAPTALDH1A1LMNAKMT2A
SCHEMBL31332780 0.77 RIPK1 (0.48) RAB9AMAPTALDH1A1LMNAKMT2A
SCHEMBL4727326 0.77 KMT2A (0.41) P2RX7RAB9AKDM4EMAPTGRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed