SCHEMBL4727593

SCHEMBL4727593

COc1cc(CC(=O)O)c2nc(C(C)(C)C)c(=O)[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.41
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
ABL1 P00519 1/20 0.41
RECQL P46063 1/20 0.41
RIN1 Q13671 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
HSD17B10 Q99714 7/20 0.41
ALDH1A1 P00352 5/20 0.39
TSHR P16473 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
AKR1C2 P52895 2/20 0.36
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
PTGS1 P23219 1/20 0.35
AKR1C3 P42330 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4660837 0.86 KDM4E (0.36) KDM4EMAPTPOLBABL1RECQL
SCHEMBL3430749 0.78 GAA (0.43) KDM4EHSD17B10GAAGRIN2DGRIN3B
SCHEMBL4662315 0.77 PTGDR2 (0.40) KDM4EMAPTPOLBABL1RECQL
SCHEMBL3353013 0.77 DHODH (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL4659621 0.74 LPAR1 (0.42) KDM4EHSD17B10ALDH1A1SMN1; SMN2AKR1C2
SCHEMBL4659631 0.70 KDM4E (0.61) KDM4EMAPTRECQLHSD17B10ALDH1A1
SCHEMBL4308637 0.70 CYP1A2 (0.52) KDM4EPOLBHSD17B10ALDH1A1TSHR
SCHEMBL3346086 0.68 PTGER4 (0.44) KDM4EGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3431673 0.68 HSD17B10 (0.41) KDM4EMAPTPOLBHSD17B10ALDH1A1
SCHEMBL4310456 0.67 ALDH1A1 (0.54) KDM4EMAPTPOLBHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008030390-A2 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION MERCK & CO., INC. (US) 2008-03-13 WO claimed
WO-2008030390-A2 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION MERCK & CO., INC. (US) 2008-03-13 WO disclosed