SCHEMBL4728129

SCHEMBL4728129

O=C1NCc2cc(OCCCCl)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
DRD2 P14416 7/20 0.42
HTR2A P28223 7/20 0.42
HTR1A P08908 6/20 0.42
KCNH2 Q12809 3/20 0.42
MAOB P27338 2/20 0.42
AURKA O14965 1/20 0.41
KDR P35968 1/20 0.41
MKNK1 Q9BUB5 2/20 0.41
SLC6A4 P31645 1/20 0.41
KCNA5 P22460 1/20 0.41
DAPK3 O43293 1/20 0.40
NTRK1 P04629 1/20 0.40
PIM1 P11309 1/20 0.40
FLT3 P36888 1/20 0.40
GSK3B P49841 1/20 0.40
ROCK1 Q13464 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4729073 0.95 DRD2 (0.43) GRM5CA12CA9DRD2HTR2A
SCHEMBL4728027 0.88 DRD2 (0.52) DRD2HTR2AHTR1AKCNH2KDR
SCHEMBL1036450 0.85 KCNA5 (0.53) GRM5DRD2MAOBKCNA5
SCHEMBL31436517 0.85 GRM5 (0.42) GRM5CA12CA9DRD2HTR2A
SCHEMBL14216502 0.85 AURKA (0.46) GRM5CA12CA9AURKAKDR
SCHEMBL4727033 0.84 DRD2 (0.53) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL14216504 0.84 MAPKAPK2 (0.45) GRM5CA12CA9DRD2HTR2A
Hydrochloric Acid SCHEMBL12503031 0.84 DAPK3 (0.43) GRM5CA12CA9DRD2HTR2A
SCHEMBL6583935 0.83 MAOB (0.47) DRD2MAOBKCNA5GSK3BHRH3
SCHEMBL26029646 0.81 TDP1 (0.43) GRM5CA12CA9AURKAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020306-A2 ISOINDOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed