SCHEMBL4729073

SCHEMBL4729073

O=C1NCc2cc(OCCCCCl)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.43
HTR2A P28223 10/20 0.43
HTR1A P08908 9/20 0.43
KCNH2 Q12809 5/20 0.43
SLC6A4 P31645 2/20 0.43
GRM5 P41594 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
MAOB P27338 1/20 0.41
AURKA O14965 1/20 0.41
KDR P35968 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
KCNA5 P22460 1/20 0.40
MAPKAPK2 P49137 1/20 0.40
DAPK3 O43293 1/20 0.40
NTRK1 P04629 1/20 0.40
PIM1 P11309 1/20 0.40
FLT3 P36888 1/20 0.40
GSK3B P49841 1/20 0.40
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728129 0.95 GRM5 (0.42) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL4727033 0.88 DRD2 (0.53) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL4728027 0.84 DRD2 (0.52) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL31436517 0.84 GRM5 (0.42) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL14216502 0.84 AURKA (0.46) GRM5CA12CA9AURKAKDR
SCHEMBL14216504 0.82 MAPKAPK2 (0.45) DRD2HTR2AHTR1AKCNH2SLC6A4
Hydrochloric Acid SCHEMBL12503031 0.82 DAPK3 (0.43) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL1036450 0.81 KCNA5 (0.53) DRD2GRM5MAOBKCNA5
SCHEMBL26029646 0.80 TDP1 (0.43) GRM5CA12CA9AURKAKDR
SCHEMBL14216501 0.80 KDM4E (0.46) GRM5CA12CA9MKNK1MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020306-A2 ISOINDOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed