SCHEMBL473103

SCHEMBL473103

CCCCOC(=O)NNCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.55
TSHR P16473 3/20 0.55
ALDH1A1 P00352 3/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
CYP3A4 P08684 1/20 0.55
MAPK1 P28482 1/20 0.55
SMN1; SMN2 Q16637 4/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
CTSK P43235 2/20 0.49
GAA P10253 1/20 0.49
RAB9A P51151 4/20 0.47
NPC1 O15118 3/20 0.47
LMNA P02545 2/20 0.47
EPHX2 P34913 1/20 0.47
RECQL P46063 1/20 0.47
POLB P06746 1/20 0.46
HPGD P15428 1/20 0.45
GLS O94925 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474570 0.94 SMN1; SMN2 (0.53) TDP1TSHRALDH1A1L3MBTL1CYP3A4
SCHEMBL9937386 0.92 SMN1; SMN2 (0.47) TDP1TSHRALDH1A1L3MBTL1CYP3A4
SCHEMBL10436016 0.85 HDAC3 (0.56) TDP1TSHRALDH1A1L3MBTL1CYP3A4
SCHEMBL14919094 0.85 MGLL (0.45) TSHRALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL3806762 0.84 EPHX2 (0.56) TDP1TSHRALDH1A1L3MBTL1CYP3A4
SCHEMBL7434407 0.84 GAA (0.60) TDP1TSHRALDH1A1MAPK1SMN1; SMN2
SCHEMBL3552049 0.81 LMNA (0.47) ALDH1A1L3MBTL1CYP3A4SMN1; SMN2CYP1A2
SCHEMBL7396978 0.80 CA12 (0.57) TDP1ALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL8800372 0.80 CYP1A2 (0.47) TDP1TSHRALDH1A1L3MBTL1CYP3A4
SCHEMBL5803249 0.80 NPC1 (0.62) TSHRALDH1A1CYP3A4MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2527297-B1 PROCESS FOR PRODUCTION OF ZINC TOLUENESULFONATE, ZINC TOLUENESULFONATE, AND PROCESS FOR PRODUCTION OF CARBAMATE MITSUI CHEMICALS INC (JP) 2018-11-21 EP disclosed
EP-2412703-B1 URETHANE COMPOUND AND PROCESS FOR PRODUCTION THEREOF, AND ISOCYANATE AND PROCESS FOR PRODUCTION THEREOF MITSUI CHEMICALS INC (JP) 2016-06-29 EP disclosed
EP-2518044-B1 METHOD FOR TREATMENT OF ISOCYANATE RESIDUE, AND METHOD FOR TREATMENT OF CARBONATE MITSUI CHEMICALS INC (JP) 2016-04-13 EP disclosed
US-9150502-B2 Urethane compound and method for producing the same, and isocyanate and method for producing the same MITSUI CHEMICALS, INC. (JP) 2015-10-06 US disclosed
US-9000219-B2 Method for treatment of isocyanate residue, and method for treatment of carbonate MITSUI CHEMICALS, INC. (JP) 2015-04-07 US disclosed
US-8664420-B2 Process for production of zinc toluenesulfonate, zinc toluenesulfonate, and process for production of carbamate MITSUI CHEMICALS, INC. (JP) 2014-03-04 US disclosed
EP-2518044-A1 METHOD FOR TREATMENT OF ISOCYANATE RESIDUE, AND METHOD FOR TREATMENT OF CARBONATE Mitsui Chemicals, Inc. (JP) 2012-10-31 EP disclosed
US-20120271067-A1 METHOD FOR TREATMENT OF ISOCYANATE RESIDUE, AND METHOD FOR TREATMENT OF CARBONATE MITSUI CHEMICALS, INC. 2012-10-25 US disclosed
US-20120259134-A1 PROCESS FOR PRODUCTION OF ZINC TOLUENESULFONATE, ZINC TOLUENESULFONATE, AND PROCESS FOR PRODUCTION OF CARBAMATE MITSUI CHEMICALS, INC. 2012-10-11 US disclosed
EP-2412703-A1 URETHANE COMPOUND AND PROCESS FOR PRODUCTION THEREOF, AND ISOCYANATE AND PROCESS FOR PRODUCTION THEREOF Mitsui Chemicals, Inc. (JP) 2012-02-01 EP disclosed
US-20120010427-A1 URETHANE COMPOUND AND METHOD FOR PRODUCING THE SAME, AND ISOCYANATE AND METHOD FOR PRODUCING THE SAME MITSUI CHEMICALS, INC. 2012-01-12 US disclosed
WO-2011076784-A2 NEW INHIBITORS OF CYCLOPHILINS AND USES THEREOF INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2011-06-30 WO disclosed
EP-0683772-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1995-11-29 EP disclosed
EP-0683772-A4 RETROVIRAL PROTEASE INHIBITING COMPOUNDS. ABBOTT LAB (US) 1995-09-27 EP disclosed
WO-1994019332-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1994-09-01 WO disclosed