SCHEMBL7434407

SCHEMBL7434407

CCOC(=O)NNCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.60
SMN1; SMN2 Q16637 4/20 0.54
PPID Q08752 1/20 0.53
MAPT P10636 4/20 0.52
LMNA P02545 3/20 0.52
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.52
HSD17B10 Q99714 2/20 0.52
HSP90AA1 P07900 1/20 0.52
HSP90AB1 P08238 1/20 0.52
APEX1 P27695 1/20 0.52
RECQL P46063 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
CYP1A2 P05177 1/20 0.49
PTGS2 P35354 1/20 0.49
NAMPT P43490 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631712 0.88 GAA (0.50) GAASMN1; SMN2PPIDMAPTLMNA
SCHEMBL7396978 0.86 CA12 (0.57) SMN1; SMN2LMNAALDH1A1TDP1NPC1
SCHEMBL473103 0.84 TDP1 (0.55) GAASMN1; SMN2LMNAALDH1A1RECQL
SCHEMBL9212256 0.83 HDAC3 (0.58) GAASMN1; SMN2MAPTLMNAALDH1A1
SCHEMBL7434290 0.83 KCNQ3 (0.53) GAASMN1; SMN2MAPTLMNAALDH1A1
Benzene SCHEMBL8878788 0.82 PPID (0.64) GAASMN1; SMN2PPIDMAPTLMNA
SCHEMBL423344 0.82 PPID (0.64) GAASMN1; SMN2PPIDMAPTLMNA
SCHEMBL2918702 0.82 GAA (0.64) GAASMN1; SMN2MAPTLMNAALDH1A1
SCHEMBL28453979 0.82 SLC26A6 (0.46) GAASMN1; SMN2LMNAKDM4ETDP1
SCHEMBL474570 0.82 SMN1; SMN2 (0.53) SMN1; SMN2LMNAALDH1A1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102695545-B Compositions comprising enzymatically cleavable ketone-modified opioid prodrugs and optional inhibitors thereof 特色疗法股份有限公司 2016-08-17 CN disclosed
CN-102917589-A Compositions comprising enzyme-cleavable opioid prodrugs and inhibitors thereof SIGNATURE THERAPEUTICS INC 2013-02-06 CN disclosed
CN-102695545-A Compositions comprising enzymatically cleavable ketone-modified opioid prodrugs and optional inhibitors thereof SIGNATURE THERAPEUTICS INC 2012-09-26 CN disclosed
EP-0640594-A1 Hydantoin derivative as metalloprotease inhibitor FUJIREBIO INC. (JP) 1995-03-01 EP disclosed