SCHEMBL4731095

SCHEMBL4731095

COCCN(C(=O)c1ccc(Cl)cc1Cl)c1cc(-c2ccc(-c3cc4ncccn4n3)cc2)sc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.36
IRAK4 Q9NWZ3 2/20 0.34
MARS1 P56192 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NPC1 O15118 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14223018 0.94 KDM4E (0.37) S1PR1IRAK4KDM4ENPSR1NPC1
SCHEMBL4730432 0.93 NPC1 (0.38) S1PR1IRAK4KDM4ENPSR1NPC1
SCHEMBL14223294 0.87 NPC1 (0.37) IRAK4KDM4ENPSR1NPC1L3MBTL1
SCHEMBL4732771 0.84 APOBEC3A (0.34) MARS1KDM4ENPC1
SCHEMBL4726531 0.81 ALDH1A1 (0.39) KDM4EALDH1A1MEN1KMT2A
SCHEMBL4726527 0.81 ALDH1A1 (0.39) KDM4EALDH1A1MEN1KMT2A
SCHEMBL4730782 0.81 IRAK4 (0.36) S1PR1IRAK4KDM4ECYP3A4
SCHEMBL4728477 0.80 SLC6A9 (0.35) IRAK4
SCHEMBL4727903 0.80 MAPT (0.39) KDM4ENPSR1NPC1KMT2A
SCHEMBL4794177 0.79 ALDH1A1 (0.37) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO claimed
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed